CI

At a glance

ClinicalIndex Comparison Record
Phase 2Completed· 55 enrolled
Drug / intervention
Temozolomide +1 moredrug
Likely dose
Temozolomide 100 mg/m² orally once daily for 7 days (then 7-day rest, repeated); R115777 400 mg orally days 8-14 and 22-28 every 4 weeksAI-extracted
Key inclusion· 8
  • Histologically proven supratentorial glioblastoma multiforme (GBM)
  • Unequivocal evidence of tumor recurrence or progression by MRI or CT scan within 14 days prior to registration
  • Stable on steroid dose for at least 5 days before imaging; new scan required if steroids increased between imaging and registration
  • Prior therapy: 0 prior chemo, OR 1 adjuvant, OR 1 adjuvant + 1 recurrent, OR 1-2 recurrent/progressive regimens
Key exclusion· 7
  • Taking CYP3A4-inducing anticonvulsants (primidone, carbamazepine, phenobarbital, phenytoin)
  • Taking drugs that interact with ZARNESTRA/R115777: cimetidine, erythromycin, azole antifungals, paclitaxel, tacrolimus, or cyclosporine
  • Uncontrolled hypertension, unstable angina, symptomatic heart failure, MI within 6 months, or serious uncontrolled cardiac arrhythmia
  • HIV positive status

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT00050986
NCT00050986Phase 2Completed

Phase I/II Evaluation Temozolomide and Farnesyl Transferase Inhibitor ZARNESTRA (R115777) for the Treatment of Recurrent and Progressive Glioblastoma Multiforme

M.D. Anderson Cancer Center·interventional·Posted Jan 3, 2003·Updated Sep 22, 2020

In Brief

A Phase 2 clinical trial evaluating Temozolomide and R115777 for Glioblastoma Multiforme. Completed, enrolled 55 participants across 1 site.

Detailed Summary

The goal of this clinical research study is to find the highest safe dose of the new drug ZARNESTRA (R115777) and temozolomide that can be given to patients with brain tumors (glioblastoma multiforme, GBM). The second goal is to learn if these drugs given in combination can shrink or slow the growth of brain tumors. The safety of this treatment will also be studied.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
CountriesUnited States
CollaboratorsJohnson & Johnson

Timeline

Phase 2CompletedFinished
2003200420052006200720082009201020112012201320142015201620172018201920202021202220232024202520262027
First PostedJan 3, 2003
Enrollment StartDec 1, 2002
Primary CompletionOct 1, 2008
TodayJul 2, 2026
Enrollment to primary: 5.8 yearsPosted 23.5 years ago

Interventions

Temozolomidedrug

Starting Dose Level: 100 mg/m\^2 taken by mouth once daily for 7 days, followed by 7 days rest and another 7-day dosing period and 7-day rest period.

R115777drug

Starting Dose Level: 400 mg taken by mouth for 7 consecutive days every other week on alternating weeks (days 8-14 and 22-28) every 4 weeks.