CI

At a glance

ClinicalIndex Comparison Record
Phase 2Completed· 140 enrolled
Drug / intervention
HKI-272 +4 moredrug
Likely dose
HKI-272 240 mgfrom record
Structured eligibility isn't available for this trial yet — see the full criteria in the Eligibility tab below.

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT01494662
NCT01494662Phase 2Completed

A Phase II Trial of HKI-272 (Neratinib), Neratinib and Capecitabine, and Ado-Trastuzumab Emtansine for Patients With Human Epidermal Growth Factor Receptor 2 (HER2)-Positive Breast Cancer and Brain Metastases

Dana-Farber Cancer Institute·interventional·Posted Dec 19, 2011·Updated Jan 23, 2026

In Brief

A Phase 2 clinical trial evaluating HKI-272, Surgical Resection, and 2 other interventions for Breast Cancer. Completed, enrolled 140 participants across 18 sites.

Detailed Summary

The purpose of this research study is to determine how well neratinib works in treating breast cancer that has spread to the brain. Neratinib is a recently discovered oral drug that may stop breast cancer cells from growing abnormally by inhibiting (or blocking) members of a family of proteins that include Human Epidermal Growth Factor Receptor 2 (HER2). In this research study, the investigators are looking to see how well neratinib works to decrease the size of or stabilize breast cancer that has spread to the brain. The investigators are also looking at how previous treatments have affected your thinking (or cognition) and how much neratinib reaches the central nervous system.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
ConditionsBreast Cancer
CountriesUnited States

Timeline

Phase 2CompletedFinished
201220132014201520162017201820192020202120222023202420252026
First PostedDec 19, 2011
Enrollment StartFeb 1, 2012
Primary CompletionFeb 1, 2023
Study CompletionApr 19, 2024
TodayJul 2, 2026
Enrollment to primary: 11 yearsPosted 14.5 years ago

Interventions

HKI-272drug

240 mg orally, once daily

Surgical Resectionprocedure

Neratinib concentrations from craniotomy specimen, CSF, plasma Neratinib.

Capecitabinedrug

750 mg/m2 orally, twice daily (1,500 mg/m2 daily) for 14 days followed by 7 days off

HKI-272drug

160 mg orally, once daily

Ado-Trastuzumab Emtansinedrug

3.6 mg/kg IV every 3 weeks