CI

At a glance

ClinicalIndex Comparison Record
Phase 1Completed· 16 enrolled
Drug / intervention
MK-3102drug
Likely dose
MK-3102 25 mg, single oral dose on Day 1AI-extracted
Key inclusion· 7
  • Chronic hepatic insufficiency lasting more than 6 months
  • Stable hepatic insufficiency with no acute episodes in the previous 2 months due to deterioration in hepatic function
  • Child-Pugh Score of 7 to 9 (moderate hepatic insufficiency)
  • Estimated creatinine clearance >60 mL/min or eGFR ≥60 mL/min/1.73 m²
Key exclusion· 8
  • History or presence of drug abuse within the past 2 years
  • History or presence of HIV
  • History or presence of hepatitis B virus (HBV) or hepatitis C virus (HCV)
  • History or presence of significant cardiovascular, pulmonary, renal, hematologic, gastrointestinal (other than hepatic impairment), endocrine, immunologic, dermatologic, or neurological disease

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT01767688
NCT01767688Phase 1Completed

An Open-Label, Single-Dose Study to Investigate the Pharmacokinetics of MK-3102 in Patients With Impaired Hepatic Function

Merck Sharp & Dohme LLC·interventional·Posted Jan 14, 2013·Updated Sep 10, 2018

In Brief

A Phase 1 clinical trial evaluating MK-3102 for Diabetes Mellitus, Type 2. Completed, enrolled 16 participants.

Detailed Summary

This study will investigate and compare the pharmacokinetics of a single 25-mg dose of MK-3102 in participants with moderate hepatic impairment and matched healthy participants. The primary hypothesis is that in participants with moderately impaired hepatic function, the area under the concentration-time curve from time zero to infinity (AUC0-∞) is similar to that observed in healthy matched control participants following a single 25 mg oral dose of MK-3102. Specifically, the true ratio (moderately impaired hepatic function patients/healthy matched control subjects) of geometric means for AUC0-∞ is no greater than 2.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
Countries--
Collaborators--

Timeline

Phase 1CompletedFinished
20132014201520162017201820192020202120222023202420252026
First PostedJan 14, 2013
Enrollment StartJan 16, 2013
Primary CompletionMar 1, 2013
Study CompletionMar 7, 2013
TodayJul 2, 2026
Enrollment to primary: 2 monthsPosted 13.5 years ago

Interventions

MK-3102drug

Single dose of 25 mg of MK-3102 (1 x 25 mg capsule) administered orally on Day 1.