CI

At a glance

ClinicalIndex Comparison Record
Phase 1Completed· 47 enrolled
Drug / intervention
XL888 +1 moredrug
Likely dose
Pembrolizumab IV and XL888 PO (specific doses not stated in criteria or arms)AI-extracted
Key inclusion· 5
  • Stage IV or locally advanced unresectable gastrointestinal adenocarcinoma (gastric, GEJ, cholangiocarcinoma, hepatocellular, pancreatic, colorectal, small intestinal) that has failed at least one prior therapy
  • For pancreatic adenocarcinoma: histologic diagnosis with locally advanced unresectable or metastatic disease failed at least one standard regimen
  • For colorectal adenocarcinoma: histologic diagnosis with locally advanced unresectable or metastatic disease; prior exposure to oxaliplatin, irinotecan, and fluoropyrimidine required
  • Measurable disease per RECIST 1.1
Key exclusion· 9
  • Prior anti-PD-1, anti-PD-L1, or anti-PD-L2 therapy
  • Prior anti-cancer monoclonal antibody within 4 weeks before study day 1 or inadequate recovery from prior agents administered >4 weeks earlier
  • Prior chemotherapy, targeted therapy, or radiation within 2 weeks of study day 1 or inadequate recovery; ≤grade 2 neuropathy allowed as exception
  • Clinically significant cardiovascular disease (MI, unstable angina within 6 months), symptomatic CHF, serious uncontrolled arrhythmia, QTc >450 msec, or prior QT prolongation with other medications

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT03095781
NCT03095781Phase 1Completed

Phase Ib Trial of Pembrolizumab and XL888 in Patients With Advanced Gastrointestinal Malignancies

Emory University·interventional·Posted Mar 30, 2017·Updated May 22, 2026

In Brief

A Phase 1 clinical trial evaluating XL888 and Pembrolizumab for Colorectal Adenocarcinoma and 14 related conditions. Completed, enrolled 47 participants across 3 sites.

Detailed Summary

This phase Ib trial studies the side effects and best dose of Hsp90 inhibitor XL888 when given together with pembrolizumab in treating patients with advanced gastrointestinal cancer that has spread to other places in the body. XL888 may stop the growth of tumor cells by blocking some of the enzymes needed for cell growth. Monoclonal antibodies, such as pembrolizumab, may block tumor growth in different ways by targeting certain cells. Giving XL888 with pembrolizumab may work better in treating patients with gastrointestinal cancer.

Study Details

Timeline

Phase 1CompletedFinished
2017201820192020202120222023202420252026
First PostedMar 30, 2017
Enrollment StartJul 7, 2017
Primary CompletionJun 10, 2021
TodayJul 2, 2026
Enrollment to primary: 3.9 yearsPosted 9.3 years ago

Interventions

XL888drug

Given PO

Pembrolizumabbiological

Given IV