CI

At a glance

ClinicalIndex Comparison Record
Phase 2Recruiting· 450 target
Drug / intervention
Fluorouracil (5-FU) +9 moredrug
Likely dose
Not stated in record
Key inclusion· 10
  • Age ≥18 years
  • Locally advanced, unresectable, or metastatic disease on recent imaging
  • Pathologically documented adenocarcinoma of stomach/GEJ/esophagus
  • HER2-positive (IHC 3+ or IHC 2+/ISH+) for Parts 1-4a
Key exclusion· 8
  • Parts 1-4: Active primary immunodeficiency, known HIV, active/past hepatitis B, hepatitis C
  • Part 5: Active uncontrolled HIV, HBV, or HCV infection
  • Uncontrolled intercurrent illness
  • History of non-infectious pneumonitis/ILD, current ILD, or suspected ILD not ruled out by imaging

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT04379596
NCT04379596Phase 2RecruitingOn Track
Long Recruiting

A Phase 1b/2 Multicenter, Open-label, Dose-escalation and Dose-expansion Study to Evaluate the Safety, Tolerability, Pharmacokinetics, Immunogenicity, and Antitumor Activity of Trastuzumab Deruxtecan (T-DXd) Monotherapy and Combinations in Adult Participants With HER2-expressing Gastric Cancer (DESTINY-Gastric-03)

AstraZeneca·interventional·Posted May 7, 2020·Updated Jun 11, 2026

In Brief

A Phase 2 clinical trial evaluating Fluorouracil (5-FU), Capecitabine, and 8 other interventions for Gastric Cancer. Currently recruiting, targeting 450 participants across 100 sites in 14 countries.

Detailed Summary

DESTINY-Gastric03 will investigate the safety, tolerability, pharmacokinetics, immunogenicity, and preliminary antitumor activity of trastuzumab deruxtecan (T-DXd) alone or in combination with chemotherapy and/or immunotherapy in HER2-expressing advanced/metastatic gastric/gastroesophageal junction (GEJ) and esophageal adenocarcinoma patients. Study hypotheses: Combination of T-DXd with cytotoxic chemotherapy and/or immunotherapy administered to subjects at the recommended phase 2 dose will show manageable safety and tolerability and preliminary anti-tumor efficacy so as to permit further clinical testing. T-DXd in combination with cytotoxic chemotherapy or immune checkpoint inhibitor administered to HER2-expressing gastric, GEJ and esophageal cancer patients who have not received prior treatment for advanced/metastatic disease will show preliminary evidence of anti-tumour activity and the potential to become a therapeutic option for this patient population.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
ConditionsGastric Cancer
CountriesBrazil, Canada, China, Germany, Italy, Japan, Netherlands, Poland, Russia, South Korea, Spain, Taiwan, United Kingdom, United States
CollaboratorsDaiichi Sankyo

Timeline

Phase 2Recruiting
2021202220232024202520262027
First PostedMay 7, 2020
Enrollment StartJun 3, 2020
Primary CompletionJun 1, 2027
TodayJul 2, 2026
Enrollment to primary: 7.0 yearsPosted 6.2 years agoPrimary completion in 11 months

Arms & Interventions

Arm 1Aexperimental

T-DXd and 5-fluorouracil (5-FU)

Drug: Fluorouracil (5-FU)Drug: Trastuzumab deruxtecan
Arm 1Bexperimental

T-DXd and capecitabine

Drug: CapecitabineDrug: Trastuzumab deruxtecan
Arm 1Cexperimental

T-DXd and durvalumab

Biological: DurvalumabDrug: Trastuzumab deruxtecan
Arm 1D(b)experimental

T-DXd, capecitabine, and oxaliplatin

Drug: CapecitabineDrug: OxaliplatinDrug: Trastuzumab deruxtecan
Arm 1E(a)experimental

T-DXd, 5-FU, and durvalumab

Drug: Fluorouracil (5-FU)Biological: DurvalumabDrug: Trastuzumab deruxtecan
Arm 1E(b)experimental

T-DXd, capecitabine, and durvalumab

Drug: CapecitabineBiological: DurvalumabDrug: Trastuzumab deruxtecan
Arm 2Aactive_comparator

Trastuzumab, 5-FU or capecitabine, and cisplatin or oxaliplatin

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: OxaliplatinBiological: TrastuzumabDrug: Cisplatin
Arm 2Bexperimental

T-DXd monotherapy

Drug: Trastuzumab deruxtecan
Arm 2Cexperimental

T-DXd, 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecan
Arm 2Dexperimental

T-DXd, pembrolizumab and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Pembrolizumab
Arm 2Eexperimental

T-DXd and pembrolizumab

Drug: Trastuzumab deruxtecanBiological: Pembrolizumab
Arm 2Fexperimental

T-DXd, pembrolizumab and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Pembrolizumab
Arm 3Aexperimental

T-DXd, Volrustomig and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Volrustomig
Arm 3Bexperimental

T-DXd, Volrustomig and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Volrustomig
Arm 4Aexperimental

T-DXd, Rilvegostomig and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Rilvegostomig
Arm 4Bexperimental

T-DXd, Rilvegostomig and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Rilvegostomig
Part 5 Main Cohortexperimental

T-DXd, Volrustomig and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Volrustomig
Part 5 Cohort 2experimental

T-DXd, Volrustomig and 5-FU or capecitabine

Drug: Fluorouracil (5-FU)Drug: CapecitabineDrug: Trastuzumab deruxtecanBiological: Volrustomig

Interventions

Fluorouracil (5-FU)drug

5-FU: administered as an IV infusion

Capecitabinedrug

Capecitabine: administered orally

Durvalumabbiological

Durvalumab: administered as an IV infusion

Oxaliplatindrug

Oxaliplatin: administered as an IV infusion

Trastuzumabbiological

Trastuzumab: administered as an IV infusion

Trastuzumab deruxtecandrug

T-DXd: administered as an IV infusion

Cisplatindrug

Cisplatin: administered as an IV infusion

Pembrolizumabbiological

Pembrolizumab: administered as an IV infusion

Volrustomigbiological

Volrustomig: administered as an IV infusion

Rilvegostomigbiological

Rilvegostomig: administered as an IV infusion