CI

At a glance

ClinicalIndex Comparison Record
Phase 2Active· 329 target
Drug / intervention
BT8009 +1 moredrug
Likely dose
Pembrolizumab 200 mgfrom record
Structured eligibility isn't available for this trial yet — see the full criteria in the Eligibility tab below.

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT04561362
NCT04561362Phase 2ActiveMonitorUpdated 7mo ago · Completion was 4mo ago
Slow Enrollment

Phase I/II Study of the Safety, Pharmacokinetics, and Preliminary Clinical Activity of BT8009 in Patients With Nectin-4 Expressing Advanced Malignancies

BicycleTx Limited·interventional·Posted Sep 23, 2020·Updated Nov 14, 2025

In Brief

A Phase 2 clinical trial evaluating BT8009 and Pembrolizumab for Urinary Bladder Neoplasm and 7 related conditions. Active but no longer recruiting, targeting 329 participants across 24 sites in 6 countries.

Signals

Enrolling slower than its timeline implies

Detailed Summary

This study is a Phase I/II, multicenter, first-in-human, open-label dose-escalation study of BT8009 given as a single agent and in combination with pembrolizumab in participants with advanced solid tumors associated with Nectin-4 expression or in participants with advanced solid tumor malignancies having renal insufficiency. The primary endpoints are: Dose limiting toxicities (Parts A-1 and A-2), Overall response rate per RECIST v1.1 (Parts B1-B7), Safety and tolerability (Parts B-8, B-9 and C), and characterization of the pharmacokinetics (Part D).

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
CountriesCanada, France, Italy, Spain, United Kingdom, United States
Collaborators--

Timeline

Phase 2Active
2021202220232024202520262027
First PostedSep 23, 2020
Enrollment StartJul 17, 2020
Primary CompletionMar 1, 2026
Study CompletionDec 1, 2026
TodayJul 2, 2026
Enrollment to primary: 5.6 yearsPosted 5.8 years ago

Interventions

BT8009drug

Bicyclic Toxin Conjugate (BTC) administered either weekly (i.e., on Days 1, 8, 15, and 22) or biweekly (Days 1 and 15) on a 28-day cycle or on Days 1 and 8 of a 21-day cycle for participants in A-1. Participants in Cohorts A-2 and B-7 will receive BT8009 weekly on 21-day cycle. Participants in Parts B-1-B-6 will receive BT8009 weekly either on a 21-day or 28-day cycle. Participants in Parts B-8 and B-9 will receive BT8009 on Days 1 and 8 of a 21-day cycle. Participants in Cohort C will receive BT8009 once weekly (i.e., on Days 1, 8, 15, and 22) on a 28-day cycle. Participants in Part D will receive BT8009 once weekly on a 28-day cycle.

Pembrolizumabdrug

Participants in Cohorts A-2 and B-7 will receive 200 mg IV over 30-minute infusion of pembrolizumab on Day 1 of each Q3W.