CI

At a glance

ClinicalIndex Comparison Record
Phase 3Completed· 566 enrolled
Drug / intervention
Xanomeline and Trospium Chloride Capsulesdrug
Likely dose
Xanomeline and Trospium Chloride Capsules 50 mgfrom record
Structured eligibility isn't available for this trial yet — see the full criteria in the Eligibility tab below.

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT04820309
NCT04820309Phase 3Completed

An Open-label Study to Assess the Long-term Safety, Tolerability, and Efficacy of KarXT in De Novo Subjects With DSM-5 Schizophrenia

Karuna Therapeutics, Inc., a Bristol Myers Squibb company·interventional·Posted Mar 29, 2021·Updated Sep 17, 2025

In Brief

A Phase 3 clinical trial evaluating Xanomeline and Trospium Chloride Capsules for Schizophrenia. Completed, enrolled 566 participants across 117 sites in 2 countries.

Detailed Summary

This is a Phase 3, multicenter, 56-week, outpatient, open-label (OL) study to evaluate the long-term safety, tolerability, and efficacy of KarXT in de novo subjects with Diagnostic and Statistical Manual-Fifth Edition (DSM-5) schizophrenia. In this OL study, all subjects will receive KarXT (a fixed combination of xanomeline 125 mg and trospium chloride 30 mg twice daily \[BID\]) for up to 52 weeks. The primary objective of the study is to assess the long-term safety and tolerability of KarXT in subjects with a DSM-5 diagnosis of schizophrenia. The secondary objective of this study is to assess the long-term efficacy and characterize the pharmacokinetics of xanomeline and trospium after administration of KarXT.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
ConditionsSchizophrenia
CountriesPuerto Rico, United States
Collaborators--

Timeline

Phase 3CompletedFinished
20222023202420252026
First PostedMar 29, 2021
Enrollment StartJun 2, 2021
Primary CompletionMay 24, 2024
TodayJul 2, 2026
Enrollment to primary: 3.0 yearsPosted 5.3 years ago

Interventions

Xanomeline and Trospium Chloride Capsulesdrug

Oral xanomeline 50 mg/trospium 20 mg BID on days 1-2 followed by xanomeline 100 mg/trospium 20 mg BID on days 3-7. The dose is increased to xanomeline 125 mg/trospium 30 mg BID on days 8-364 unless the subject is experiencing adverse events from the xanomeline 100 mg/ trospium 20 mg dose. Subjects who were increased to xanomeline 125 mg/trospium 30 mg will have the option to return to xanomeline 100 mg/ trospium 20 mg depending on clinical response and tolerability. Re-escalation to 125/30 BID or re-titration in cases in which the subject has been off KarXT for a longer period of time (at least a week) is allowed and will require a discussion between the principal investigator and the medical monitor.