CI

At a glance

ClinicalIndex Comparison Record
Phase 3Active· 373 enrolled / 373 target
Drug / intervention
Giredestrant +6 moredrug
Likely dose
Giredestrant 30 milligramsfrom record
Structured eligibility isn't available for this trial yet — see the full criteria in the Eligibility tab below.

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT05306340
NCT05306340Phase 3ActiveUpdate Overdue (7.9/mo)Completion was 11mo ago

A Phase III, Randomized, Open-Label, Multicenter Study Evaluating the Efficacy and Safety of Giredestrant Plus Everolimus Compared With the Physician's Choice of Endocrine Therapy Plus Everolimus in Patients With Estrogen Receptor-Positive, HER2-Negative, Locally Advanced or Metastatic Breast Cancer

Genentech, Inc.·interventional·Posted Apr 1, 2022·Updated Jun 17, 2026

In Brief

A Phase 3 clinical trial evaluating Giredestrant, Exemestane, and 5 other interventions for Estrogen Receptor (ER)-Positive, HER2-negative, Locally Advanced or Metastatic Breast Cancer. Active but no longer recruiting, targeting 373 participants across 136 sites in 13 countries.

Signals

Enrollment appears stalled

Detailed Summary

This Phase III, randomized, open-label, multicenter study will evaluate the efficacy and safety of giredestrant plus everolimus compared with the physician's choice of endocrine therapy plus everolimus in participants with estrogen receptor (ER)-positive, human epidermal growth factor receptor 2 (HER2)-negative locally advanced or metastatic breast cancer who have had previous treatment with cyclin-dependent kinase 4/6 inhibitors (CDK4/6is) and endocrine therapy, either in the locally advanced/metastatic or the adjuvant setting.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
CountriesArgentina, Germany, Greece, Italy, Japan, Singapore, South Africa, South Korea, Spain, Taiwan, Turkey (Türkiye), United Kingdom, United States
Collaborators--

Timeline

Phase 3Active
2023202420252026
First PostedApr 1, 2022
Enrollment StartAug 3, 2022
Primary CompletionJul 16, 2025
Study CompletionOct 15, 2026
TodayJul 2, 2026
Enrollment to primary: 3.0 yearsPosted 4.3 years ago

Arms & Interventions

Giredestrant plus Everolimusexperimental

Drug: GiredestrantDrug: EverolimusDrug: LHRH AgonistDrug: Dexamethasone Mouth Rinse
Physician's Choice of Endocrine Therapy plus Everolimusactive_comparator

The physician's choice of endocrine therapy is defined as either exemestane, fulvestrant, or tamoxifen.

Drug: ExemestaneDrug: FulvestrantDrug: TamoxifenDrug: EverolimusDrug: LHRH AgonistDrug: Dexamethasone Mouth Rinse

Interventions

Giredestrantdrug

Participants will receive treatment with giredestrant 30 milligrams (mg) orally once a day (QD) on Days 1-28 of each 28-day cycle until unacceptable toxicity or disease progression as determined by the investigator according to Response Evaluation Criteria in Solid Tumors, version 1.1 (RECIST v1.1).

Exemestanedrug

If exemestane is chosen as the physician's choice of endocrine therapy, the participant will receive exemestane at a dose of 25 mg orally once a day (QD) on Days 1-28 of each 28-day cycle or as per local label, until unacceptable toxicity or disease progression as determined by investigator according to RECIST v1.1.

Fulvestrantdrug

If fulvestrant is chosen as the physician's choice of endocrine therapy, the participant will receive fulvestrant in the clinic at a dose of 500 mg intramuscularly on Day 1 and Day 15 of Cycle 1, then Day 1 of each cycle thereafter (1 cycle is 28 days) or as per local prescribing information, until unacceptable toxicity or disease progression as determined by investigator according to RECIST v1.1.

Tamoxifendrug

If tamoxifen is chosen as the physician's choice of endocrine therapy, the participant will receive tamoxifen at a dose of 20 mg orally QD on Days 1-28 of each 28-day cycle or as per local prescribing information, until unacceptable toxicity or disease progression as determined by investigator according to RECIST v1.1.

Everolimusdrug

Participants will receive treatment with everolimus 10 mg orally QD during each 28-day cycle until unacceptable toxicity or disease progression as determined by the investigator according to RECIST v1.1.

LHRH Agonistdrug

Only premenopausal/perimenopausal female participants and male participants will receive a luteinizing hormone-releasing hormone (LHRH) agonist on Day 1 of each 28-day treatment cycle. The investigator will determine and supply the appropriate LHRH agonist locally approved for use in breast cancer.

Dexamethasone Mouth Rinsedrug

A compounded alcohol-free mouthwash of dexamethasone (0.5 mg in 5 mL) will be supplied, where feasible. It is strongly recommended for prophylaxis or treatment of stomatitis/mucositis. Participants should use the alcohol-free mouthwash of dexamethasone four times QD for 8 weeks started concurrently with study treatment, and use it reactively thereafter with the first appearance of symptoms.