CI

At a glance

ClinicalIndex Comparison Record
Phase 1Recruiting· 320 target
Drug / intervention
Divarasib +4 moredrug
Likely dose
Pembrolizumab 200 mgfrom record
Key inclusion· 6
  • Confirmation of Biomarker eligibility
  • ECOG performance status 0 or 1
  • Histologically or cytologically documented locally advanced unresectable or metastatic NSCLC not eligible for curative surgery and/or definitive chemoradiotherapy
  • No prior systemic treatment for advanced unresectable or metastatic NSCLC
Key exclusion· 11
  • Known concomitant second oncogenic driver with available targeted treatment
  • Squamous cell histology NSCLC
  • Symptomatic, untreated, or actively progressing CNS metastases (Cohorts A, B, and C)
  • Prior treatment with a KRAS G12C inhibitor

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

In the news

1 article

Matched to this trial by ClinicalIndexfrom reputable biotech & medical press.

Search/NCT05789082
NCT05789082Phase 1RecruitingHigh Momentum
Long Recruiting

A Phase Ib/II, Open-Label, Multicenter Study Evaluating the Safety, Activity, and Pharmacokinetics of Divarasib as a Single Agent or in Combination With Other Anti-Cancer Therapies in Patients With Previously Untreated Advanced Or Metastatic Non-Small Cell Lung Cancer With a KRAS G12C Mutation

Hoffmann-La Roche·interventional·Posted Mar 29, 2023·Updated Jun 15, 2026

In Brief

A Phase 1 clinical trial evaluating Divarasib, Pembrolizumab, and 3 other interventions for Non-Small Cell Lung Cancer. Currently recruiting, targeting 320 participants across 71 sites in 18 countries.

Signals

Enrolling ahead of pace

Detailed Summary

The purpose of this study is to evaluate the safety, pharmacokinetics (PK), and activity of single-agent divarasib or combined with other anti-cancer therapies in participants with previously untreated, advanced or metastatic non-small cell lung cancer (NSCLC).

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
CountriesArgentina, Australia, Belgium, Brazil, Canada, China, Israel, Italy, Japan, Netherlands, Poland, South Korea, Spain, Sweden, Switzerland, Taiwan, United Kingdom, United States
Collaborators--

Timeline

Phase 1Recruiting
2023202420252026202720282029203020312032
First PostedMar 29, 2023
Enrollment StartJun 20, 2023
Primary CompletionJan 29, 2032
TodayJul 2, 2026
Enrollment to primary: 8.6 yearsPosted 3.3 years agoPrimary completion in 5.6 years

Arms & Interventions

Cohort A - Combination Dose Finding + Dose Expansionexperimental

Participants will be enrolled in different cohorts to receive divarasib (different dose levels will be evaluated) once a day (QD) combined with pembrolizumab 200 mg intravenous (IV) infusion every 3 weeks (Q3W). During the expansion stage, some participants are planned to be randomized to one divarasib combination dose level; other participants are planned to be randomized to another divarasib combination dose level. Divarasib will be given in combination with pembrolizumab.

Drug: DivarasibDrug: Pembrolizumab
Cohort B - Combination Dose Finding + Dose Expansionexperimental

Participants enrolled in this cohort will receive divarasib (different dose levels will be evaluated) QD combined with pembrolizumab 200 mg IV Q3W plus investigator's choice of platinum-based chemotherapy (carboplatin or cisplatin) and pemetrexed.

Drug: DivarasibDrug: PembrolizumabDrug: CarboplatinDrug: CisplatinDrug: Pemetrexed
Cohort C - Dose Expansionexperimental

Participants enrolled in this cohort will receive one dose level of divarasib QD.

Drug: Divarasib
Cohort D - Dose Expansionexperimental

Participants enrolled in this cohort will receive one dose level of divarasib QD.

Drug: Divarasib

Interventions

Divarasibdrug

Participants will receive divarasib orally (PO), QD on days 1-21 of each 21-day cycle.

Pembrolizumabdrug

Participants will receive a 200 mg IV infusion of pembrolizumab Q3W on Day 1 of each 21-day cycle.

Carboplatindrug

Participants will receive IV carboplatin Q3W for four 21-day cycles.

Cisplatindrug

Participants will receive IV cisplatin Q3W for four 21-day cycles.

Pemetrexeddrug

Participants will receive IV pemetrexed Q3W.