CI

At a glance

ClinicalIndex Comparison Record
Phase 1Completed· 50 enrolled
Drug / intervention
Orforglipron +6 moredrug
Likely dose
Not stated in record
Structured eligibility isn't available for this trial yet — see the full criteria in the Eligibility tab below.

Standardized by ClinicalIndex from the ClinicalTrials.gov record · verify against the source.

Search/NCT06186622
NCT06186622Phase 1Completed

A Drug-Drug Interaction Study to Assess the Effect of Orforglipron on the Pharmacokinetics of Digoxin, Simvastatin, Rosuvastatin, Acetaminophen, and Midazolam in Healthy Overweight and Obese Participants

Eli Lilly and Company·interventional·Posted Jan 2, 2024·Updated May 22, 2026

In Brief

A Phase 1 clinical trial evaluating Orforglipron, Simvastatin, and 5 other interventions for Healthy and 2 related conditions. Completed, enrolled 50 participants across 2 sites.

Detailed Summary

The main purpose of this study is to determine effect of orforglipron capsule formulation on the amount of digoxin, rosuvastatin, acetaminophen, midazolam, and simvastatin (each given alone and together with orforglipron) that enters the bloodstream and how long it takes the body to eliminate them when administered orally in healthy overweight and obese participants. In addition, the effect of the orforglipron tablet on the amount of simvastatin that enters the bloodstream and how long it takes the body to eliminate it will be evaluated. The study will also assess the effect of sodium bicarbonate when administered alone with simvastatin versus orforglipron capsule containing sodium bicarbonate administered with simvastatin. The safety and tolerability of orforglipron and information about any side effects experienced will be collected. Study will be conducted in two parts, with part 1 and 2 lasting up to approximately 23 and 24 weeks each, including the screening period.

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
CountriesUnited States
Collaborators--

Timeline

Phase 1CompletedFinished
202420252026
First PostedJan 2, 2024
Enrollment StartJan 2, 2024
Primary CompletionJul 10, 2024
TodayJul 2, 2026
Enrollment to primary: 6 monthsPosted 2.5 years ago

Interventions

Orforgliprondrug

Administered orally.

Simvastatindrug

Administered orally.

Digoxindrug

Administered orally.

Rosuvastatindrug

Administered orally.

Acetaminophendrug

Administered orally.

Midazolamdrug

Administered orally.

Sodium Bicarbonatedrug

Administered orally.