CI

At a glance

ClinicalIndex Comparison Record
N/ACompleted· 30 enrolled
Drug / intervention
Estradiol (E2) +1 moredrug
Likely dose
Estradiol (E2) 2 mgfrom record
Structured eligibility isn't available for this trial yet — see the full criteria in the Eligibility tab below.

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Search/NCT07145281
NCT07145281N/ACompleted

Comparing the Effects of Sublingual Estradiol Treatment Versus Oral Estradiol With Cyproterone Acetate (CPA) Treatment on The Coagulation System in Transgender Women: A Prospective, Controlled Cohort Study

Tel-Aviv Sourasky Medical Center·interventional·Posted Aug 28, 2025·Updated Aug 28, 2025

In Brief

A clinical study evaluating Estradiol (E2) and Cyproterone Acetate (Androcur, BAY94-8367) for Gender Dysphoria, Adult and 5 related conditions. Completed, enrolled 30 participants across 1 site.

Detailed Summary

The goal of this clinical trial is to learn about the effects of different routes of estradiol administration on blood clotting in transgender women starting gender-affirming hormone therapy. The main questions it aims to answer are: Does sublingual estradiol reduce free Protein S levels compared to oral estradiol with cyproterone acetate? Does sublingual estradiol accelerate activation of the clotting system, as measured by thrombin generation? Researchers will compare sublingual estradiol to oral estradiol plus cyproterone acetate to see if the way estradiol is taken changes blood clotting risk. Participants will: Take either sublingual estradiol (2 mg daily in divided doses) or oral estradiol (2 mg daily) with cyproterone acetate (10 mg daily) for 6 months Provide blood samples at baseline and after 6 months to measure hormone levels and clotting factors Attend clinic visits for monitoring, including safety checks and routine laboratory tests

Study Details

Study Typeinterventional
Allocation--
Masking--
Primary Purpose--
CountriesIsrael
Collaborators--

Timeline

N/ACompletedFinished
2023202420252026
First PostedAug 28, 2025
Enrollment StartNov 10, 2022
Primary CompletionNov 10, 2024
TodayJul 2, 2026
Enrollment to primary: 2 yearsPosted 10 months ago

Interventions

Estradiol (E2)drug

Participants receive estradiol 2 mg/day. In the experimental arm, estradiol is administered sublingually in four divided doses (0.5 mg each). In the active comparator arm, estradiol is administered orally, in combination with cyproterone acetate, for 6 months. All participants are treatment-naive.

Cyproterone Acetate (Androcur, BAY94-8367)drug

Participants in the active comparator arm receive cyproterone acetate (CPA) 10 mg orally, once daily, in combination with oral estradiol, for 6 months. All participants are treatment-naive.